COURSE UNIT TITLE

: DRUG SYNTHESIS

Description of Individual Course Units

Course Unit Code Course Unit Title Type Of Course D U L ECTS
KIM 4259 DRUG SYNTHESIS ELECTIVE 2 0 0 3

Offered By

Chemistry

Level of Course Unit

First Cycle Programmes (Bachelor's Degree)

Course Coordinator

PROFESSOR DOCTOR MUSTAFA YAVUZ ERGÜN

Offered to

Chemistry

Course Objective

The aim of this course is to inform students about structure, nomenclature, reactions and synthesis of heterocyclic compounds.

Learning Outcomes of the Course Unit

1   At the end of this course students will have information about structure and classification of nonheterocyclic drugs
2   At the end of this course students will have information about synthesis of nonheterocyclic drugs
3   At the end of this course students will be able to understand structure and clssification of heterocyclic drugs
4   At the end of this course students will be able to understand synthesis of heterocyclic drugs
5   At the end of this course students will have information about synthesis of active ingredients of drugs.

Mode of Delivery

Face -to- Face

Prerequisites and Co-requisites

None

Recomended Optional Programme Components

None

Course Contents

Week Subject Description
1 Aliphatic and Alicyclic Drugs
2 Monocyclic Aromatic Drugs
3 Polycyclic Aromatic Drugs
4 Steroids
5 Five Membered Ring Heterocyclic Drugs
6 Six Membered Ring Heterocyclic Drugs
7 Five Membered Ring Benzofused Heterocyclic Drugs
8 Six Membered Ring Benzofused Heterocyclic Drugs
9 Bicyclic Fused Heterocyclic Drugs
10 -Lactam Antibiotics
11 Miscellaneous Heterocyclic Drugs and Alkaloids
12 Homework presentation
13 Homework presentation
14 Homework presentation

Recomended or Required Reading

Textbook(s):
1. Organic Chemistry of Drug Synthesis, D. Lednicer, L. A. Mitscher, G. I. Georg, John Wiley&sons, Inc., 1990.

Supplementary Book(s):
1. Heterocyclic Chemistry, J. A. Joule, G. F. Smith, Redwood Burn Limited, 1976.

Planned Learning Activities and Teaching Methods

Presentation, Lecture, question and answer technique, homework, examples

Assessment Methods

SORTING NUMBER SHORT CODE LONG CODE FORMULA
1 MTE MIDTERM EXAM
2 ASG ASSIGNMENT
3 FIN FINAL EXAM
4 FCGR FINAL COURSE GRADE (RESIT) MTE * 0.25 + ASG * 0.25 + FIN * 0.50
5 RST RESIT
6 FCGR FINAL COURSE GRADE (RESIT) MTE * 0.25 + ASG * 0.25 + RST * 0.50


Further Notes About Assessment Methods

None

Assessment Criteria

Student will be evaluated with homework presentation and final exam. Homework presentations will be made during the last three weeks of the semester.

Language of Instruction

Turkish

Course Policies and Rules

To continue 70% of the classes throughout the semester is students own responsibility. The specified class times must be complied with. Unethical behavior that may occur in class and on exams, will be acting within the framework of the relevant regulations. D.E.U. Science Faculty implementation principles of teaching and examination regulations can be found at http://web.deu.edu.tr/fen

Contact Details for the Lecturer(s)

D.E.U. Science Faculty Department of Chemistry
e-mail: yavuz.ergun@deu.edu.tr

Office Hours

To be announced.

Work Placement(s)

None

Workload Calculation

Activities Number Time (hours) Total Work Load (hours)
Lectures 11 2 22
Preparation for midterm exam 1 10 10
Preparation for final exam 1 20 20
Preparing presentations 1 20 20
Final 1 2 2
Midterm 1 1 1
TOTAL WORKLOAD (hours) 75

Contribution of Learning Outcomes to Programme Outcomes

PO/LOPO.1PO.2PO.3PO.4PO.5PO.6PO.7PO.8PO.9PO.10PO.11PO.12PO.13PO.14PO.15PO.16PO.17
LO.1321422
LO.2321422
LO.3321422
LO.4321422
LO.5321422